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| Place of Origin: | China |
| Brand Name: | Pharmlab |
| Certification: | ISO 9001, USP,GMP |
| Model Number: | 168273-06-1 |
| Minimum Order Quantity: | negotiation |
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| Price: | negotiation |
| Packaging Details: | Disguised package ; Foil bag |
| Delivery Time: | 3-5 work days |
| Payment Terms: | Western Union, MoneyGram, T/T, bitcoin |
| Supply Ability: | Mass in stock |
| Product Name: | Rimonabant | CAS: | 168273-06-1 |
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| Appearance: | White Crystalline Powder | Usage: | Weight Loss |
| Same Products: | DXM, DNP | Contact Person: | Betty |
| High Light: | topical anesthetic drugs,pain killer powder |
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Rimonabant hydrochloride (SR-141716A) is a potent and selective CB1 inverse agonist/antagonist with a Ki of 1.6 nM, minimal affinity for CB2, and and some GPR55 agonist activity. Rimonabant was developed as an anti-obesity drug because of its appetite suppressant activity, but was taken off the market because of side effects of depression and anxiety.
Rimonabant works by blocking endogenous binding to neuronal CB1 receptors. Activation of these receptors by endoegenous , such as anadamide, increases appetite. It is the most advanced receptor antagonist in clinical development and offers a novel therapeutic approach to appetite control and weight reduction.
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Product Name |
Rimonabant |
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CAS |
168273-06-1 |
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Melting point |
230 to 240 |
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Molecular Formula |
C22Cl3HN4O |
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Dry weight loss |
less than 0.5% |
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PH |
(10% aqueous solution) 4-7 |
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Heavy metal |
less than 10ppm |
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TLC |
only one spot |
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Content |
99.5% |
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Character |
white or white crystalline powder, soluble in methanol. |
Rimonabant is the new weight-loss drug, can be applied to smoking cessation. A new weight-loss drug rimonabant (Rimonabant), not only can lose weight, but also lower blood pressure, cholesterol and blood sugar, domestically year clinical study found that subjects taking one to two months later, weight average minus six to eight kilograms.
As well as keeping you lean, the drug also helps you quit the smoking habit. This will be of great interest for many smokers who are afraid to give up because they say they will put on loads of weight if they do (young female smokers worry about this the most).
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Product Name |
Rimonabant |
Batch No. |
170928 |
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Report Date |
2017/09/28 |
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Test Items |
Specification |
Test Results |
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Appearance |
Off white crystalline powder |
Off white crystalline powder |
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Melting Point |
233.2℃~236.1℃ |
230℃~240℃ |
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L.O.D |
0.23% |
<0.5% |
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Solubility |
Conforms |
Freely soluble in methanol |
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Heavy metals(Pb) |
10ppm |
<10ppm |
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Assay |
99.65% |
>99.5% |
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T.L.C. |
Only one spot |
Only one spot |
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1) Rimonabant(Acomplia) was studied to be used complementary to diet and exercise to treat obese or overweight patients who suffer from type 2 diabetes and abnormal levels of fat in the blood.
2) Sanofi argued that Acomplia could also prevent the risk of cardiovascular disease.
Patients with large waist circumference (102 cm in men and 88 cm in women) were said to most benefit from taking the drug.
3) Smoking cessation
Rimonabant may also be found to be effective in assisting some smokers to quit smoking. first, to use rimonabant directly to aid in smoking cessation; second, to help prevent weight gain in former smokers.
It is expected that the usual dose of rimonabant will be 20 mg once daily before breakfast. No dosage adjustment is recommended for the elderly, but this agent should be used with caution in patients older than 75 years of age.
Although rimonabant can be used in patients with mild hepatic impairment, caution is advised in patients with moderate impairment. This medication is not recommended for those with severe hepatic impairment.
Rimonabant may be used cautiously in patients with mild-to-moderate renal impairment, but it is not recommended for patients who are severely renally impaired.
There are no data supporting the use of rimonabant in pediatric populations.
Rimonabant should not be given to patients with a known hypersensitivity to the agent or any compound found in the tablet formulation.
The drug is contraindicated in lactat-ing women and is not recommended for use in women who are pregnant.
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24/7 online for problems and concern related to the product |
Contact Person: Coco
Tel: +8618186204104
